{"id":1479,"date":"2021-07-21T13:07:22","date_gmt":"2021-07-21T11:07:22","guid":{"rendered":"https:\/\/fjarno.org\/revista-renal\/?p=1479"},"modified":"2021-07-21T13:07:22","modified_gmt":"2021-07-21T11:07:22","slug":"curiositats-la-ciclosporina","status":"publish","type":"post","link":"https:\/\/fjarno.org\/revista-renal\/curiositats-la-ciclosporina\/","title":{"rendered":"Curiositats, La Ciclosporina."},"content":{"rendered":"<p><b>Sabies qu\u00e8&#8230;?<\/b><\/p>\n<p><span style=\"font-weight: 400;\">La ciclosporina \u00e9s un f\u00e0rmac immunosupressor d&#8217;acci\u00f3 r\u00e0pida i efica\u00e7. \u00c9s un f\u00e0rmac cl\u00e0ssicament utilitzat per evitar el rebuig en individus sotmesos a trasplantaments d&#8217;\u00f2rgans.\u00a0<\/span><\/p>\n<p><b>Els or\u00edgens<\/b><\/p>\n<p><span style=\"font-weight: 400;\">La hist\u00f2ria de la ciclosporina s&#8217;inicia en l&#8217;any 1969 partint d&#8217;una mostra de terra d\u2019una regi\u00f3 del sud de Noruega. D&#8217;aquesta mostra de terra s&#8217;a\u00eflla un fong, Tolypocladium inflatum Gams, del qual s&#8217;extreuen dues subst\u00e0ncies que mostren una activitat anti-f\u00fangica i antibi\u00f2tica residual, insuficient per pensar en qualsevol aplicaci\u00f3 farmac\u00e8utica. No obstant aix\u00f2, tenint en compte la m\u00ednima toxicitat d&#8217;aquestes subst\u00e0ncies, es va decidir realitzar un cribratge farmacol\u00f2gic a la recerca de possibles aplicacions terap\u00e8utiques.\u00a0<\/span><\/p>\n<p><span style=\"font-weight: 400;\">Les subst\u00e0ncies de l&#8217;extracte del fong inhibien la formaci\u00f3 d&#8217;anticossos, sense impedir la multiplicaci\u00f3 de les c\u00e8l\u00b7lules leuc\u00e8miques inoculades en ratolins. La troballa (1972) era sorprenent: es tractava de subst\u00e0ncies capaces d&#8217;inhibir la resposta immunit\u00e0ria, per\u00f2 no bloquejant la proliferaci\u00f3 cel\u00b7lular. Com a m\u00ednim, aquestes subst\u00e0ncies podrien ser molt valuoses com a eina de recerca.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">El 1980, un grup d&#8217;investigadors de Sandoz, dirigit per R. Wenger, va aconseguir la s\u00edntesi de la mol\u00e8cula al laboratori. (1)<\/span><\/p>\n<p><b>Ciclosporina i covid-19<\/b><\/p>\n<p><span style=\"font-weight: 400;\">Segons un estudi realitzat pel Grup de Recerca en la COVID-19, liderat pel Servei de Medicina Interna de l&#8217;Hospital Universitari Quir\u00f3nsalud Madrid, juntament amb la Universitat Europea, la Ciclosporina sembla ser un f\u00e0rmac prometedor per a pacients hospitalitzats per la Covid-19. Els pacients que van rebre ciclosporina van tenir un 81 per cent menys de probabilitat de morir que els pacients que no van rebre aquest tractament.<\/span><\/p>\n<p><span style=\"font-weight: 400;\">El Dr. Daniel Carnevali, cap de Servei de Medicina Interna de l&#8217;Hospital Universitari Quir\u00f3nsalud Madrid i professor de la Universitat Europea admet que tot i els resultats semblen prometedors, per confirmar aquesta hip\u00f2tesi caldria un assaig cl\u00ednic en el qual es pogu\u00e9s aleatoritzar entre pacients que prenguessin ciclosporina o placebo &#8220;. (2)<\/span><\/p>\n<p>&nbsp;<\/p>\n<ol>\n<li style=\"font-weight: 400;\" aria-level=\"1\"><span style=\"font-weight: 400;\">L\u00f3pez, J.M (2 de mar\u00e7 de 2019). <\/span><i><span style=\"font-weight: 400;\">Ciclosporina: un hito de la farmacolog\u00eda de los trasplantes<\/span><\/i><span style=\"font-weight: 400;\">. Info-Farmacia. Recuperado el 16 de julio de 2021 de <\/span><a href=\"http:\/\/www.info-farmacia.com\/medico-farmaceuticos\/revisiones-farmaceuticas\/hitos-de-la-farmacologia-ciclosporina\"><span style=\"font-weight: 400;\">http:\/\/www.info-farmacia.com\/medico-farmaceuticos\/revisiones-farmaceuticas\/hitos-de-la-farmacologia-ciclosporina<\/span><\/a><\/li>\n<\/ol>\n<p><span style=\"font-weight: 400;\">\u00a0Sanitaria 2000 S.L (17 de novembre de 2020). <\/span><i><span style=\"font-weight: 400;\">Ciclosporina, un f\u00e1rmaco prometedor para pacientes hospitalizados por la Covid-19<\/span><\/i><span style=\"font-weight: 400;\">.\u00a0 Sanidadprivada.com. Recuperat el 16 de juliol de 2021 de <\/span><a href=\"http:\/\/sanidadprivada.publicacionmedica.com\/noticia\/ciclosporina-un-farmaco-prometedor-para-pacientes-hospitalizados-por-la-covid-19\"><span style=\"font-weight: 400;\">http:\/\/sanidadprivada.publicacionmedica.com\/noticia\/ciclosporina-un-farmaco-prometedor-para-pacientes-hospitalizados-por-la-covid-19<\/span><\/a><\/p>\n","protected":false},"excerpt":{"rendered":"<p>Sabies qu\u00e8&#8230;? La ciclosporina \u00e9s un f\u00e0rmac immunosupressor d&#8217;acci\u00f3 r\u00e0pida i efica\u00e7. \u00c9s un f\u00e0rmac cl\u00e0ssicament utilitzat per evitar el rebuig en individus sotmesos a trasplantaments d&#8217;\u00f2rgans.\u00a0 Els or\u00edgens La hist\u00f2ria de la ciclosporina s&#8217;inicia en l&#8217;any 1969 partint d&#8217;una mostra de terra d\u2019una regi\u00f3 del sud de Noruega. D&#8217;aquesta mostra de terra s&#8217;a\u00eflla un [&hellip;]<\/p>\n","protected":false},"author":3,"featured_media":1481,"comment_status":"open","ping_status":"open","sticky":false,"template":"","format":"standard","meta":{"footnotes":""},"categories":[13,11],"tags":[34],"class_list":{"0":"post-1479","1":"post","2":"type-post","3":"status-publish","4":"format-standard","5":"has-post-thumbnail","7":"category-curiositats","8":"category-salut-ciencia","9":"tag-numero-4"},"yoast_head":"<!-- This site is optimized with the Yoast SEO plugin v27.5 - https:\/\/yoast.com\/product\/yoast-seo-wordpress\/ -->\n<title>Curiositats, La Ciclosporina. | Revista Renal<\/title>\n<meta name=\"robots\" content=\"index, follow, max-snippet:-1, max-image-preview:large, max-video-preview:-1\" \/>\n<link rel=\"canonical\" href=\"https:\/\/fjarno.org\/revista-renal\/curiositats-la-ciclosporina\/\" \/>\n<meta property=\"og:locale\" content=\"ca_ES\" \/>\n<meta property=\"og:type\" content=\"article\" \/>\n<meta property=\"og:title\" content=\"Curiositats, La Ciclosporina. | Revista Renal\" \/>\n<meta property=\"og:description\" content=\"Sabies qu\u00e8&#8230;? 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